Tranexamic acid is a prescription drug to treat melasma
Tranexamic Acid is very often prescribed to treat heavy periods and is deemed safe by the FDA. It is not yet FDA-approved for the treatment of melasma. Despite that, doctors prescribe it very often to treat melasma.
We do not fully understand how tranexamic acid works for melasma. But it may work by inhibiting an enzyme called tyrosinase that produces the brown pigment melanin in your skin. This pigment causes the brownish colour of melasma. Approximately 89% of women who take tranexamic acid report that their melasma fades.